dc.contributor.author |
Smolobochkin A.V. |
|
dc.contributor.author |
Turmanov R.A. |
|
dc.contributor.author |
Abdullaeva D.S. |
|
dc.contributor.author |
Gazizov A.S. |
|
dc.contributor.author |
Voronina J.K. |
|
dc.contributor.author |
Appazov N.O. |
|
dc.contributor.author |
Buzyurova D.N. |
|
dc.contributor.author |
Burilov A.R. |
|
dc.contributor.author |
Pudovik M.A. |
|
dc.date.accessioned |
2021-02-25T20:56:25Z |
|
dc.date.available |
2021-02-25T20:56:25Z |
|
dc.date.issued |
2020 |
|
dc.identifier.uri |
https://dspace.kpfu.ru/xmlui/handle/net/162748 |
|
dc.description.abstract |
© 2020 Wiley-VCH GmbH A first successful synthesis of 2-(het)aryl-N-phosphorylpyrrolidines is reported starting from readily available N-(4,4-diethoxybutyl)amides of P(V) acids. A range of phenols and hydroxyl-substituted O-heterocycles may be employed into the reaction furnishing N-phosphorylated 2-(het)arylpyrrolidines with up to 90 % yield. The developed method permits a presence of sensitive to phosphorylation hydroxy groups and provides the easy and regioselective entry to target compounds. |
|
dc.subject |
Cyclization |
|
dc.subject |
Nitrogen heterocycles |
|
dc.subject |
Phosphorus amides |
|
dc.subject |
Pyrrolidines |
|
dc.subject |
Synthetic methods |
|
dc.title |
2-(Het)aryl-N-phosphorylpyrrolidines via Cyclization of Phosphorus Acid Amides: A Regioselective Approach |
|
dc.type |
Article |
|
dc.relation.ispartofseries-issue |
39 |
|
dc.relation.ispartofseries-volume |
5 |
|
dc.collection |
Публикации сотрудников КФУ |
|
dc.relation.startpage |
12045 |
|
dc.source.id |
SCOPUS-2020-5-39-SID85093828882 |
|