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Browsing by Author "Lenina O.A."

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6-Methyluracil derivatives as peripheral site ligand-hydroxamic acid conjugates: Reactivation for paraoxon-inhibited acetylcholinesterase

Semenov V.E.; Zueva I.V.; Lushchekina S.V.; Lenina O.A.; Gubaidullina L.M.; Saifina L.F.; Shulaeva M.M.; Kayumova R.M.; Saifina A.F.; Gubaidullin A.T.; Kondrashova S.A.; Latypov S.K.; Masson P.; Petrov K.A. (2020)

© 2019 Elsevier Masson SAS New uncharged conjugates of 6-methyluracil derivatives with imidazole-2-aldoxime and 1,2,4-triazole-3-hydroxamic acid units were synthesized and studied as reactivators of organophosphate-inhibited ...
Cationic liposomes mediated transdermal delivery of meloxicam and ketoprofen: Optimization of the composition, in vitro and in vivo assessment of efficiency

Kuznetsova D.A.; Vasileva L.A.; Gaynanova G.A.; Vasilieva E.A.; Lenina O.A.; Nizameev I.R.; Kadirov M.K.; Petrov K.A.; Zakharova L.Y.; Sinyashin O.G. (2021)

New liposomes modified with pyrrolidinium surfactants containing a hydroxyethyl fragment (CnPB, n = 12, 14, 16) were prepared for transdermal delivery of non-steroidal anti-inflammatory drugs. In order to obtain the optimal ...
Modulation of aggregation behavior, antimicrobial properties and catalytic activity of piperidinium surfactants by modifying their head group with a polar fragment

Kushnazarova R.A.; Mirgorodskaya A.B.; Kuznetsov D.M.; Tyryshkina A.A.; Voloshina A.D.; Gumerova S.K.; Lenina O.A.; Nikitin E.N.; Zakharova L.Y. (2021)

To establish the effect of surfactants structure on their functional activity a number of alkyl-N-hydroxyethylpiperidinium bromides with different length of the hydrophobic tail were synthesized and characterized. Aggregation ...
Novel acetylcholinesterase inhibitors based on uracil moiety for possible treatment of Alzheimer disease

Semenov V.E.; Zueva I.V.; Mukhamedyarov M.A.; Lushchekina S.V.; Petukhova E.O.; Gubaidullina L.M.; Krylova E.S.; Saifina L.F.; Lenina O.A.; Petrov K.A. (2020)

© 2020 by the authors In this study, novel derivatives based on 6-methyluracil and condensed uracil were synthesized, namely, 2,4-quinazoline-2,4-dione with ω-(ortho-nitrilebenzylethylamino) alkyl chains at the N atoms of ...
Slow-binding reversible inhibitor of acetylcholinesterase with long-lasting action for prophylaxis of organophosphate poisoning

Lenina O.A.; Zueva I.V.; Zobov V.V.; Semenov V.E.; Masson P.; Petrov K.A. (2020)

© 2020, The Author(s). Organophosphorus (OP) compounds represent a serious health hazard worldwide. The dominant mechanism of their action results from covalent inhibition of acetylcholinesterase (AChE). Standard therapy ...
Water-soluble betaines and amines based on thiacalix[4]arene scaffold as new cholinesterase inhibitors

Padnya P.L.; Bayarashov E.E.; Zueva I.V.; Lushchekina S.V.; Lenina O.A.; Evtugyn V.G.; Osin Y.N.; Petrov K.A.; Stoikov I.I. (2020)

© 2019 Elsevier Inc. Novel ammonium and betaine derivatives of p-tert-butylthiacalix[4]arene in cone and 1,3-alternate conformation were synthesized with high yields for the first time. The obtained compounds form in water ...

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Browsing by Author "Lenina O.A."

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