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Просмотр по автору "Sapozhnikov S.V."

Просмотр по автору "Sapozhnikov S.V."

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  • Sapozhnikov S.V.; Sabirova A.E.; Shtyrlin N.V.; Druk A.Y.; Agafonova M.N.; Chirkova M.N.; Kazakova R.R.; Grishaev D.Y.; Nikishova T.V.; Krylova E.S.; Nikitina E.V.; Kayumov A.R.; Shtyrlin Y.G. (2021)
    A diverse series of 43 novel “soft antimicrobials” based on quaternary ammonium pyridoxine derivatives which include six-membered acetals and ketals of pyridoxine bound via cleavable linker moieties (amide, ester) with a ...
  • Shtyrlin N.V.; Pugachev M.V.; Sapozhnikov S.V.; Garipov M.R.; Vafina R.M.; Grishaev D.Y.; Pavelyev R.S.; Kazakova R.R.; Agafonova M.N.; Iksanova A.G.; Lisovskaya S.A.; Zeldi M.I.; Krylova E.S.; Nikitina E.V.; Sabirova A.E.; Kayumov A.R.; Shtyrlin Y.G. (2020)
    © 2020 by the authors. A series of 108 novel quaternary bis-ammonium pyridoxine derivatives carrying various substituents at the quaternary nitrogen’s and acetal carbon was synthesized. Thirteen compounds exhibited ...
  • Sapozhnikov S.V.; Pavelyev R.S.; Shtyrlin N.V.; Shtyrlin Y.G. (2021)
    In this work we have described the transformation of synthetic route of the antiseptic drug candidate Pyridosept. Initial method has included in seven steps and has poor overall yield of target compound. This is the ...

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